1-(2-Nitrophenyl)thiosemicarbazides: A novel class of potent, orally active non-peptide antagonist for the bradykinin B2 receptor [2]

Edward K. Dziadulewicz; Timothy J. Ritchie; Allan Hallett; Christopher R. Snell; Soo Y. Ko; Roger Wrigglesworth; Glyn A. Hughes; Andrew R. Dunstan; Graham C. Bloomfield; Gillian S. Drake; Michael C. Brown; Wai Lee; Gillian M. Burgess; Clare Davis; Mohammed Yaqoob; Martin N. Perkins; Elizabeth A. Campbell; Andrew J. Davis; Humphrey P. Rang

doi:10.1021/jm991155o

1-(2-Nitrophenyl)thiosemicarbazides: A novel class of potent, orally active non-peptide antagonist for the bradykinin B₂ receptor [2]

Edward K. Dziadulewicz
, Timothy J. Ritchie
, Allan Hallett
, Christopher R. Snell
, Soo Y. Ko
, Roger Wrigglesworth
, Glyn A. Hughes
, Andrew R. Dunstan
, Graham C. Bloomfield
, Gillian S. Drake
, Michael C. Brown
, Wai Lee
, Gillian M. Burgess
, Clare Davis
, Mohammed Yaqoob
, Martin N. Perkins
, Elizabeth A. Campbell
, Andrew J. Davis
, Humphrey P. Rang

Department of Chemistry & Nanoscience

Research output: Contribution to journal › Letter › peer-review

30 Scopus citations

Original language	English
Pages (from-to)	769-771
Number of pages	3
Journal	Journal of Medicinal Chemistry
Volume	43
Issue number	5
DOIs	https://doi.org/10.1021/jm991155o
State	Published - 9 Mar 2000

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10.1021/jm991155o

Cite this

Dziadulewicz, E. K., Ritchie, T. J., Hallett, A., Snell, C. R., Ko, S. Y., Wrigglesworth, R., Hughes, G. A., Dunstan, A. R., Bloomfield, G. C., Drake, G. S., Brown, M. C., Lee, W., Burgess, G. M., Davis, C., Yaqoob, M., Perkins, M. N., Campbell, E. A., Davis, A. J., & Rang, H. P. (2000). 1-(2-Nitrophenyl)thiosemicarbazides: A novel class of potent, orally active non-peptide antagonist for the bradykinin B₂ receptor [2]. Journal of Medicinal Chemistry, 43(5), 769-771. https://doi.org/10.1021/jm991155o

@article{1b5f6a84106f4b4e87da46b59f9a2cb0,

title = "1-(2-Nitrophenyl)thiosemicarbazides: A novel class of potent, orally active non-peptide antagonist for the bradykinin B2 receptor [2]",

author = "Dziadulewicz, \{Edward K.\} and Ritchie, \{Timothy J.\} and Allan Hallett and Snell, \{Christopher R.\} and Ko, \{Soo Y.\} and Roger Wrigglesworth and Hughes, \{Glyn A.\} and Dunstan, \{Andrew R.\} and Bloomfield, \{Graham C.\} and Drake, \{Gillian S.\} and Brown, \{Michael C.\} and Wai Lee and Burgess, \{Gillian M.\} and Clare Davis and Mohammed Yaqoob and Perkins, \{Martin N.\} and Campbell, \{Elizabeth A.\} and Davis, \{Andrew J.\} and Rang, \{Humphrey P.\}",

year = "2000",

month = mar,

day = "9",

doi = "10.1021/jm991155o",

language = "English",

volume = "43",

pages = "769--771",

journal = "Journal of Medicinal Chemistry",

issn = "0022-2623",

publisher = "American Chemical Society",

number = "5",

}

Dziadulewicz, EK, Ritchie, TJ, Hallett, A, Snell, CR, Ko, SY, Wrigglesworth, R, Hughes, GA, Dunstan, AR, Bloomfield, GC, Drake, GS, Brown, MC, Lee, W, Burgess, GM, Davis, C, Yaqoob, M, Perkins, MN, Campbell, EA, Davis, AJ & Rang, HP 2000, '1-(2-Nitrophenyl)thiosemicarbazides: A novel class of potent, orally active non-peptide antagonist for the bradykinin B₂ receptor [2]', Journal of Medicinal Chemistry, vol. 43, no. 5, pp. 769-771. https://doi.org/10.1021/jm991155o

TY - JOUR

T1 - 1-(2-Nitrophenyl)thiosemicarbazides

T2 - A novel class of potent, orally active non-peptide antagonist for the bradykinin B2 receptor [2]

AU - Dziadulewicz, Edward K.

AU - Ritchie, Timothy J.

AU - Hallett, Allan

AU - Snell, Christopher R.

AU - Ko, Soo Y.

AU - Wrigglesworth, Roger

AU - Hughes, Glyn A.

AU - Dunstan, Andrew R.

AU - Bloomfield, Graham C.

AU - Drake, Gillian S.

AU - Brown, Michael C.

AU - Lee, Wai

AU - Burgess, Gillian M.

AU - Davis, Clare

AU - Yaqoob, Mohammed

AU - Perkins, Martin N.

AU - Campbell, Elizabeth A.

AU - Davis, Andrew J.

AU - Rang, Humphrey P.

PY - 2000/3/9

Y1 - 2000/3/9

UR - https://www.scopus.com/pages/publications/0034624707

U2 - 10.1021/jm991155o

DO - 10.1021/jm991155o

M3 - Letter

C2 - 10715143

AN - SCOPUS:0034624707

SN - 0022-2623

VL - 43

SP - 769

EP - 771

JO - Journal of Medicinal Chemistry

JF - Journal of Medicinal Chemistry

IS - 5

ER -